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Development of novel fluorescent histamine H₁-receptor antagonists to study ligand-binding kinetics in living cells (2018)
Journal Article
antagonists to study ligand-binding kinetics in living cells. Scientific Reports, 8, doi:10.1038/s41598-018-19714-2. ISSN 2045-2322

The histamine H1-receptor (H1R) is an important mediator of allergy and inflammation. H1R antagonists have particular clinical utility in allergic rhinitis and urticaria. Here we have developed six novel fluorescent probes for this receptor that are... Read More